One-Pot Synthesis of 2,3-Dihydro-pyrrolopyridinones Using in Situ Generated Formimines - Normandie Université Access content directly
Journal Articles Organic Letters Year : 2007

One-Pot Synthesis of 2,3-Dihydro-pyrrolopyridinones Using in Situ Generated Formimines

Abstract

A novel one-pot methodology is described for the synthesis of functionalized pyrrolopyridinones using in situ generated formimines and an ortho-lithiated pyridinecarboxamide species. Depending on the reaction conditions, this procedure allows versatile access to aminomethylated pyridinecarboxamides, 2,3-dihydro-pyrrolopyridinones, or 1,1-dialkylated 2,3-dihydro-pyrrolopyridinone derivatives.

Dates and versions

hal-02385488 , version 1 (28-11-2019)

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Geoffrey Deguest, Laurent Bischoff. One-Pot Synthesis of 2,3-Dihydro-pyrrolopyridinones Using in Situ Generated Formimines. Organic Letters, 2007, 9 (3), pp.545-545. ⟨10.1021/ol063033d⟩. ⟨hal-02385488⟩
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