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Journal Articles Beilstein Journal of Organic Chemistry Year : 2017

Synthesis of the heterocyclic core of the D-series GE2270

Abstract

A straightforward enantiomerically pure synthesis of the heterocyclic core of the D-series GE2270 is reported. The synthetic strategy combines the Hantzsch thiazole’s building condensation with a cross-coupling reaction including direct C–H hetarylation to build and connect step-by-step thiazolyl moieties to the 5-bromopicolinate as readily available starting material.

Dates and versions

hal-02046259 , version 1 (22-02-2019)

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Christophe Berini, Thibaut Martin, Pierrik Lassalas, Francis Marsais, Christine Baudequin, et al.. Synthesis of the heterocyclic core of the D-series GE2270. Beilstein Journal of Organic Chemistry, 2017, 13, pp.1407-1412. ⟨10.3762/bjoc.13.137⟩. ⟨hal-02046259⟩
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