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Potent 3‐Hydroxy‐2‐Pyridine Aldoxime Reactivators of Organophosphate‐Inhibited Cholinesterases with Predicted Blood–Brain Barrier Penetration
Tamara Zorbaz
,
Anissa Braïki
,
Nikola Marakovic
,
Julien Renou
,
Eugenio de La Mora
,
et al.
Journal articles
hal-02024542v1
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Reactivators of acetylcholinesterase inhibited by organophosphorus nerve agents
Guillaume Mercey
,
Tristan Verdelet
,
Julien Renou
,
Maria Kliachyna
,
Rachid Baati
,
et al.
Journal articles
hal-01015972v1
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Design, synthesis and biological evaluation of novel tetrahydroacridine pyridine- aldoxime and -amidoxime hybrids as efficient uncharged reactivators of nerve agent-inhibited human acetylcholinesterase
Maria Kliachyna
,
Gianluca Santoni
,
Valentin Nussbaum
,
Julien Renou
,
Benoît Sanson
,
et al.
Journal articles
hal-01131268v1
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Synthesis and in vitro and in vivo evaluations of New Uncharged reactivators for cholinesterases inhibited by organophosphorus nerve agents
Anissa Braïki
,
Julien Renou
,
Romain Mougeot
,
Florian Nachon
,
José Dias
,
et al.
Medical Chemical Defense Conference (MCDC, 17, 2019), Mar 2019, Munich, Germany
Conference poster
hal-02543452v1
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Tryptoline-3-hydroxypyridinaldoxime conjugates as efficient reactivators of phosphylated human acetyl and butyrylcholinesterase
Julien Renou
,
Melanie Loiodice
,
Melanie Arboleas
,
Rachid Baati
,
Ludovic Jean
,
et al.
Journal articles
hal-01150284v1
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Syntheses and in vitro evaluations of uncharged reactivators for human acetylcholinesterase inhibited by organophosphorus nerve agents.
Julien Renou
,
Guillaume Mercey
,
Tristan Verdelet
,
Emilia Păunescu
,
Emilie Gillon
,
et al.
Journal articles
hal-00996535v1
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Synthesis and in vitro evaluation of donepezil-based reactivators and analogues for nerve agent-inhibited human acetylcholinesterase
Julien Renou
,
José Dias
,
Guillaume Mercey
,
Tristan Verdelet
,
Catherine Rousseau
,
et al.
Journal articles
hal-02046237v1
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Uncharged reactivators of cholinesterases inhibited by organophosphorus nerve agents.
Nicolas Probst
,
Anissa Braïki
,
Pierre Warnault
,
Julien Renou
,
Catherine Gomez
,
et al.
International Meeting on Cholinesterases (13, 2018) and International Conference on Paraoxonases (7, 2018)), Sep 2018, Hradec Králové, Czech Republic
Conference poster
hal-02543467v1
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New Uncharged reactivators for cholinesterases inhibited by organophosphorus nerve agents
Anissa Braïki
,
Julien Renou
,
Romain Mougeot
,
Tamara Zorbaz
,
André-Guilhem Calas
,
et al.
International Conference on Chemical Biological Radiological nuclear Explosive - Research & Innovation (CBRNE, 2, 2017), May 2017, Lyon, France
Conference poster
hal-02544823v1
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Design and Development of New Uncharged Reactivators of OP-Inhibited Cholinesterases
Pierre Warnault
,
Julien Renou
,
Catherine Gomez
,
Guillaume Mercey
,
Tristan Verdelet
,
et al.
International Conference on Chemical Biological Radiological and Nuclear agents (CBRN) - Research & Innovation (1, 2015), Mar 2015, Antibes, France
Conference poster
hal-02544917v1
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Phenyltetrahydroisoquinoline-pyridinaldoxime conjugates as efficient uncharged reactivators for the dephosphylation of inhibited human acetylcholinesterase.
Guillaume Mercey
,
Julien Renou
,
Tristan Verdelet
,
Maria Kliachyna
,
Rachid Baati
,
et al.
Journal articles
hal-00996512v1
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A miniaturized peptidyl-prolyl isomerase enzyme assay
Mirella Vivoli
,
Julien Renou
,
Arnaud Chevalier
,
Isobel H. Norville
,
Suraya Diaz
,
et al.
Journal articles
hal-02046314v1
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Synthesis and evaluations of uncharged reactivators for cholinesterases inhibited by organophosphate agents
Anissa Braïki
,
Julien Renou
,
Romain Mougeot
,
Florian Nachon
,
André-Guilhem Calas
,
et al.
International Conference on Chemical Biological Radiological and Nuclear agents (CBRN) - Research & Innovation (3, 2019), May 2019, Nantes, France
Conference poster
hal-02543439v1
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Novel uncharged reactivators against OP-inhibition of human acetylcholinesterase
Rachid Baati
,
Maria Klyachina
,
Valentin Nussbaum
,
Pierre-Yves Renard
,
Ludovic Jean
,
et al.
France, Patent n° : EP13306584.7. 2013
Patents
hal-01150304v1
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Synthesis of new uncharged reactivators for cholinesterases inhibited by organophosphorus nerve agents
Anissa Braïki
,
Julien Renou
,
Catherine Gomez
,
Romain Mougeot
,
Florian Nachon
,
et al.
Tetrahedron Symposium (17, 2016), Jun 2016, Barcelone, Spain
Conference poster
hal-02544884v1
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Uncharged Reactivators of cholinesterases Inhibited by organophosphorus nerve agents
Pierre Warnault
,
Julien Renou
,
Catherine Gomez
,
Guillaume Mercey
,
Tristan Verdelet
,
et al.
International Meeting on Cholinesterases - Sixth International Conference on Paraoxonases (12, 2015), Sep 2015, Elche, Spain
Conference poster
hal-02544902v1
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